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Nancy E Kohl Selected Research

compound 30

10/2021Discovery of 6-[(3S,4S)-4-Amino-3-methyl-2-oxa-8-azaspiro[4.5]decan-8-yl]-3-(2,3-dichlorophenyl)-2-methyl-3,4-dihydropyrimidin-4-one (IACS-15414), a Potent and Orally Bioavailable SHP2 Inhibitor.
7/2008Kinesin spindle protein (KSP) inhibitors. 9. Discovery of (2S)-4-(2,5-difluorophenyl)-n-[(3R,4S)-3-fluoro-1-methylpiperidin-4-yl]-2-(hydroxymethyl)-N-methyl-2-phenyl-2,5-dihydro-1H-pyrrole-1-carboxamide (MK-0731) for the treatment of taxane-refractory cancer.

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Nancy E Kohl Research Topics

Disease

14Neoplasms (Cancer)
10/2021 - 07/2003
2Non-Small-Cell Lung Carcinoma (Carcinoma, Non-Small Cell Lung)
11/2020 - 03/2007
2Hepatocellular Carcinoma (Hepatoma)
12/2019 - 04/2015
2Precursor Cell Lymphoblastic Leukemia-Lymphoma (Acute Lymphoblastic Leukemia)
05/2015 - 04/2009
1Sarcoma (Soft Tissue Sarcoma)
10/2021
1Nausea
12/2019
1Diarrhea
12/2019
1Vomiting
12/2019
1Glioblastoma (Glioblastoma Multiforme)
02/2016
1Prostatic Neoplasms (Prostate Cancer)
06/2015
1Acute Myeloid Leukemia (Acute Myelogenous Leukemia)
05/2015
1Ewing Sarcoma (Sarcoma, Ewing)
05/2013
1Stomach Neoplasms (Stomach Cancer)
02/2010
1Primary Myelofibrosis (Myelosclerosis)
08/2009
1Essential Thrombocythemia
08/2009
1Polycythemia (Erythrocytosis)
08/2009
1Polycythemia Vera
08/2009
1Precursor T-Cell Lymphoblastic Leukemia-Lymphoma (T-ALL)
04/2009
1Colonic Neoplasms (Colon Cancer)
09/2008
1Neoplasm Metastasis (Metastasis)
03/2007
1Lung Neoplasms (Lung Cancer)
03/2007
1Carcinoma (Carcinomatosis)
04/2006

Drug/Important Bio-Agent (IBA)

2Receptor Protein-Tyrosine Kinases (Tyrosine Kinase Receptors)IBA
10/2021 - 02/2010
2compound 30IBA
10/2021 - 07/2008
2LigandsIBA
02/2016 - 02/2010
2Protein-Tyrosine Kinases (Tyrosine Kinase)IBA
05/2013 - 08/2009
2Small Interfering RNA (siRNA)IBA
05/2013 - 03/2007
2Phosphotransferases (Kinase)IBA
05/2013 - 03/2005
2Proteins (Proteins, Gene)FDA Link
07/2008 - 03/2005
1Mitogen-Activated Protein KinasesIBA
10/2021
1Phosphoric Monoester Hydrolases (Phosphatases)IBA
10/2021
1Tyrosine Kinase InhibitorsIBA
11/2020
1osimertinibIBA
11/2020
1fisogatinibIBA
12/2019
1Immune Checkpoint ProteinsIBA
02/2016
1Immune Checkpoint InhibitorsIBA
02/2016
1AntibodiesIBA
02/2016
1N- (4- methyl- 3- (1- methyl- 7- (6- methylpyridin- 3- ylamino)- 2- oxo- 1,2- dihydropyrimido(4,5- d)pyrimidin- 3(4H)- yl)phenyl)- 3- (trifluoromethyl)benzamideIBA
05/2015
1Fibroblast Growth Factors (Fibroblast Growth Factor)IBA
04/2015
1BLU9931IBA
04/2015
1Messenger RNA (mRNA)IBA
04/2015
1Type 4 Fibroblast Growth Factor ReceptorIBA
04/2015
1Focal Adhesion Protein-Tyrosine KinasesIBA
05/2013
1PF-562271IBA
05/2013
1Tyrosine (L-Tyrosine)FDA Link
05/2013
1Phosphatidylinositols (Phosphatidylinositol)IBA
02/2010
1Extracellular Signal-Regulated MAP Kinases (Extracellular Signal Regulated Kinases)IBA
02/2010
15H- benzo(4,5)cyclohepta(1,2- b)pyridin- 5- oneIBA
02/2010
1ErythropoietinFDA Link
08/2009
1Janus Kinase 2IBA
08/2009
1Notch ReceptorsIBA
04/2009
1Amyloid Precursor Protein Secretases (beta-Secretase)IBA
04/2009
1Gamma Secretase Inhibitors and ModulatorsIBA
04/2009
1Fatty Acids (Saturated Fatty Acids)IBA
09/2008
1EnzymesIBA
09/2008
1KinesinsIBA
07/2008
1taxaneIBA
07/2008
1Cytotoxins (Cytolysins)IBA
07/2008
1PyrrolesIBA
07/2008
1AminesIBA
05/2007
1ErbB Receptors (EGF Receptor)IBA
03/2007
1Intercellular Signaling Peptides and Proteins (Growth Factors)IBA
03/2007
1Hepatocyte Growth Factor (Growth Factor, Hepatocyte)IBA
03/2007
1Urea (Carbamide)FDA LinkGeneric
04/2006
1pyrrolineIBA
04/2006
1AmidesIBA
04/2006
1Biomarkers (Surrogate Marker)IBA
03/2005
1geranylgeranyltransferase type-I (protein geranylgeranyltransferase)IBA
07/2003
1p21(ras) farnesyl-protein transferase (protein farnesyltransferase)IBA
07/2003

Therapy/Procedure

9Therapeutics
10/2021 - 03/2005
1Intravenous Injections
06/2015
1Castration
06/2015